Compile Data Set for Download or QSAR
maximum 50k data
Found 75 of ec50 data for polymerid = 50003158
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50601513(CHEMBL5180351)
Affinity DataEC50:  37nMAssay Description:Agonist activity at rat KCNQ2 channel expressed in CHO cells by patch clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65882(2-[(5-fluoro-3-nitro-1H-indol-2-yl)thio]acetic aci...)
Affinity DataEC50:  170nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65903(4-butyl-N-[2-(2-furanyl)-2-(4-morpholinyl)ethyl]-1...)
Affinity DataEC50:  920nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65904(1-[1-(1,3-benzodioxol-5-yl)ethyl]-3-(2-ethoxypheny...)
Affinity DataEC50:  1.51E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65902(5-chloranyl-2-[(3-methylphenyl)methylsulfonyl]-N-(...)
Affinity DataEC50:  1.83E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65905(3-(4-tert-butylphenoxy)-N-(2-morpholin-4-yl-2-thio...)
Affinity DataEC50:  1.97E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50143558(CHEMBL41355 | EZOGABINE | N-(2-amino-4-(4-fluorobe...)
Affinity DataEC50:  2.04E+3nMAssay Description:Agonist activity at rat KCNQ2 channel expressed in CHO cells by patch clamp methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65889(1-[(2,2-dichlorocyclopropyl)methyl]-3-(4-methylphe...)
Affinity DataEC50:  2.17E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM50143558(CHEMBL41355 | EZOGABINE | N-(2-amino-4-(4-fluorobe...)
Affinity DataEC50:  2.17E+3nMAssay Description:Agonist activity at rat KCNQ2 expressed in CHOK1 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65922(1-(2,4-dichlorobenzyl)-3-phenyl-urea | 1-[(2,4-dic...)
Affinity DataEC50:  2.22E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65947(1-(6-chloranylpyridin-3-yl)-3-(3-fluorophenyl)urea...)
Affinity DataEC50:  2.81E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65894(5-chloranyl-2-[(3-methylphenyl)methylsulfonyl]-N-(...)
Affinity DataEC50:  2.89E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65880(MLS000529853 | S-[2-[(6-fluoranyl-3-prop-2-ynyl-1,...)
Affinity DataEC50:  2.97E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65879(2-(dimethylcarbamoylthiocarbamoylamino)-4-(5-methy...)
Affinity DataEC50:  3.01E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65890(5-chloranyl-2-[(4-methylphenyl)methylsulfonyl]-N-(...)
Affinity DataEC50:  3.02E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65883(2-chloranyl-5-[(2Z)-2-(2-oxidanylidene-1-propan-2-...)
Affinity DataEC50:  3.70E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65944(1-(6-chloranylpyridin-3-yl)-3-[(2,4-dichlorophenyl...)
Affinity DataEC50:  3.74E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65949(1-(6-bromanylpyridin-3-yl)-3-(3-fluorophenyl)urea ...)
Affinity DataEC50:  4.04E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65901(5-chloranyl-2-[(2-fluorophenyl)methylsulfonyl]-N-(...)
Affinity DataEC50:  4.19E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65931(1-(3-chloranyl-4-fluoranyl-phenyl)-3-pyridin-3-yl-...)
Affinity DataEC50:  4.21E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65886(1-(4-phenoxyphenyl)-3-(3-pyridinyl)thiourea | 1-(4...)
Affinity DataEC50:  4.45E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM64280(5-chloranyl-2-[(4-fluorophenyl)methylsulfonyl]-N-(...)
Affinity DataEC50:  4.47E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65899(5-chloranyl-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[(...)
Affinity DataEC50:  4.80E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65881(2-(4-chloro-2-methyl-5-{[4-(2-pyridinyl)-1-piperaz...)
Affinity DataEC50:  5.34E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65897(5-chloranyl-2-[(4-methylphenyl)methylsulfonyl]-N-(...)
Affinity DataEC50:  5.40E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65946(1-(3-fluorophenyl)-3-(6-fluoro-3-pyridinyl)urea | ...)
Affinity DataEC50:  5.76E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM64871(N-(6-chloranylpyridin-3-yl)-4-fluoranyl-benzamide ...)
Affinity DataEC50:  5.80E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Mode of Action, Electrophysiology Source (MLPCN Center Name): Johns Hopkins Ion Channel...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM64871(N-(6-chloranylpyridin-3-yl)-4-fluoranyl-benzamide ...)
Affinity DataEC50:  5.90E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Mode of Action, Electrophysiology Source (MLPCN Center Name): Johns Hopkins Ion Channel...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65898(2-benzylsulfonyl-5-chloro-N-(5-isopropyl-1,3,4-thi...)
Affinity DataEC50:  6.20E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65923(1-(3-Fluoro-phenyl)-3-pyridin-3-yl-urea | 1-(3-flu...)
Affinity DataEC50:  6.28E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65943(1-(2,4-dichlorobenzyl)-3-(6-fluoro-3-pyridyl)urea ...)
Affinity DataEC50:  6.31E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65951(1-(3-fluorophenyl)-3-(5-fluoro-3-pyridinyl)urea;2,...)
Affinity DataEC50:  6.32E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65948(1-(6-bromanyl-5-methyl-pyridin-3-yl)-3-(3-fluoroph...)
Affinity DataEC50:  6.61E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65926(1-(4-chlorophenyl)-3-(3-pyridinyl)urea | 1-(4-chlo...)
Affinity DataEC50:  6.85E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65270(MLS000705220 | N'-(5-bromo-3-chloro-2-hydroxyb...)
Affinity DataEC50:  7.13E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65886(1-(4-phenoxyphenyl)-3-(3-pyridinyl)thiourea | 1-(4...)
Affinity DataEC50:  7.25E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM63846((4-Chloro-phenyl)-(6-chloro-pyridazin-3-yl)-amine ...)
Affinity DataEC50:  7.86E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65900(5-chloranyl-2-[(2-fluorophenyl)methylsulfonyl]-N-(...)
Affinity DataEC50:  8.40E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65945(1-(2,4-dichlorobenzyl)-3-(5-fluoro-3-pyridyl)urea;...)
Affinity DataEC50:  8.64E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65934(1-(3-fluoranyl-4-methyl-phenyl)-3-pyridin-3-yl-ure...)
Affinity DataEC50:  9.14E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65935(1-(3-chlorophenyl)-3-(3-pyridinyl)thiourea | 1-(3-...)
Affinity DataEC50:  9.33E+3nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM48038(4-[(E)-[3-(2-methylanilino)-4-oxo-1-naphthalenylid...)
Affinity DataEC50:  9.51E+3nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65941(1-(3,5-dimethylphenyl)-3-(3-pyridinyl)urea | 1-(3,...)
Affinity DataEC50:  1.07E+4nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65933(1-(4-anilinophenyl)-3-(3-pyridinyl)thiourea | 1-(4...)
Affinity DataEC50:  1.10E+4nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65885(MLS001000844 | N-(4-methyl-2-nitro-phenyl)-2-pheny...)
Affinity DataEC50:  1.14E+4nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65877((6E)-2,4-bis(chloranyl)-6-[(1,3-thiazol-2-ylamino)...)
Affinity DataEC50:  1.16E+4nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65878(MLS000547588 | N-(4-naphthalen-2-yloxyphenyl)furan...)
Affinity DataEC50:  1.20E+4nMAssay Description:BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65950(1-(3-fluorophenyl)-3-(5-methyl-3-pyridinyl)urea;2,...)
Affinity DataEC50:  1.24E+4nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65936(1-(3-pyridyl)-3-(4-sec-butylphenyl)thiourea | 1-(4...)
Affinity DataEC50:  1.26E+4nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetPotassium voltage-gated channel subfamily KQT member 2(Rattus norvegicus)
Shanghai Institute Of Materia Medica

Curated by ChEMBL
LigandPNGBDBM65940(1-(3,4-dimethylphenyl)-3-(3-pyridinyl)urea | 1-(3,...)
Affinity DataEC50:  1.35E+4nMAssay Description:Name: Dose response of Retigabine-insensitive compounds that potentiate KCNQ2 potassium channel BioAssay Type: Confirmatory, Concentration-Response R...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
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